Norflurazepam 10 MG Pellets Product Description

Introduction

Norflurazepam, also known as N-Desalkylflurazepam or 2-oxoquazepam, is an active metabolite of several benzodiazepines such as flurazepam, flutoprazepam, and quazepam. It exhibits strong anxiolytic, sedative, muscle relaxant, and anticonvulsant properties. Norflurazepam 10 mg pellets provide a precise, convenient dosage form designed for research purposes, allowing controlled studies on benzodiazepine pharmacology and toxicology.

Chemical Properties and Specifications

Structural and Molecular Characteristics

• Chemical Formula: C15H10ClFN2O

• Molecular Weight: 288.70 g/mol

• CAS Number: 2886-65-9

• IUPAC Name: 7-chloro-5-(2-fluorophenyl)-2,3-dihydro-1H-1,4-benzodiazepin-2-one

• Synonyms: Norflurazepam, N-desalkylflurazepam, 2-oxoquazepam

Physical Properties and Formulation

• Appearance: White to off-white solid pellets

• Purity: High-grade research standard (>98%)

• Dosage Per Pellet: 10 mg of Norflurazepam

• Packaging: Typically blister packs or vials ensuring precise dosing and protection

Pharmacological Profile and Mechanism of Action

• Acts as a positive allosteric modulator of the GABA-A receptor

• Produces sedative, anxiolytic, muscle relaxant, and anticonvulsant effects

• Long elimination half-life (47-150 hours) contributing to sustained effects and accumulation potential

Research Applications

• Laboratory investigations into benzodiazepine metabolism and pharmacodynamics

• Forensic toxicology for benzodiazepine identification and quantification

• Behavioral pharmacology and receptor binding studies

Safety and Handling

• Use personal protective equipment (gloves, eye protection) during handling

• Handle in ventilated laboratory conditions to reduce exposure risk

• Follow hazardous chemical disposal regulations

Regulatory Status

• Controlled substance in many regions, regulated as a benzodiazepine derivative

• Strictly for use in scientific and forensic research only

• Verify compliance with local laws prior to acquisition and use

Frequently Asked Questions (FAQs)

1. What is the dosage in one pellet?
   Each pellet contains exactly 10 mg of Norflurazepam.

2. What are the effects of Norflurazepam?
   Sedative, anxiolytic, muscle relaxant, and anticonvulsant effects typical of benzodiazepines.

3. How should pellets be stored?
   Store in a cool, dry, and dark environment.

4. Is Norflurazepam approved for human use?
   No, for research purposes only.

5. What is its half-life?
   Between 47 and 150 hours, leading to long-effect duration.

Conclusion

Norflurazepam 10 mg pellets provide a stable, accurately dosed research chemical for studying benzodiazepine pharmacology, metabolism, and forensic toxicology. Proper safety precautions and regulatory compliance are mandatory for laboratory use.