Flubrotizolam 0.5 MG Fanax Bars Product Description

Introduction

Flubrotizolam 0.5 mg Fanax Bars are precise dosage forms containing 0.5 milligrams of the active compound Flubrotizolam, a potent thienotriazolodiazepine class benzodiazepine analog. These bars are designed for reliable dosing in pharmacological and neuroscientific research studying GABA-A receptor modulation and central nervous system depression. Flubrotizolam is known for its sedative, anxiolytic, and muscle relaxant effects.

Chemical Properties and Specifications

2.1 Structural and Molecular Characteristics

• Chemical Formula: C17H12BrFN4S

• Molecular Weight: 377.24 g/mol

• CAS Number: 57801-95-3

• IUPAC Name: 2-bromo-4-(2-fluorophenyl)-9-methyl-6H-thieno[3,2-f]triazolo[4,3-a]diazepine

• Synonyms: Flubrotizolam, Fanax Bars

2.2 Physical Properties and Pellet Specifications

• Appearance: Solid bar form, white to off-white, approximately 8mm diameter

• Dosage: 0.5 mg active Flubrotizolam per bar

• Purity: ≥98% pharmaceutical/research grade

• Storage Recommendations: Store in a cool, dry, dark place within airtight packaging to maintain stability for up to two years

Pharmacological Profile and Mechanism of Action

3.1 Mechanism of Action

Flubrotizolam is a potent positive allosteric modulator at GABA-A receptors, particularly at benzodiazepine binding sites. It enhances the effect of GABA, the primary inhibitory neurotransmitter in the CNS, resulting in sedation, anxiolysis, muscle relaxation, and anticonvulsant effects. Its chemical structure imparts high receptor affinity and potency.

3.2 Research Applications

Widely used for research into benzodiazepine receptor pharmacodynamics and CNS pharmacology. The bar format allows for precise dosing crucial in controlled experimental models of CNS depression, sedation, and anxiety regulation.

Comparative Analysis with Related Compounds

4.1 Comparison with Other Benzodiazepines

Flubrotizolam has a higher potency and longer action profile compared to traditional benzodiazepines like alprazolam or diazepam. It offers enhanced binding due to its thienotriazolodiazepine framework with bromine and fluorine substitutions, useful for studying high-affinity benzodiazepine interactions.

4.2 Advantages for Research

Fanax bars are convenient for dosing and reduce dosing errors compared to powder forms. The 0.5 mg dosage per bar is optimal for a variety of in vivo and in vitro research protocols.

Safety and Handling Guidelines

5.1 Laboratory Safety

Use appropriate PPE, including gloves and eye protection. Handle in well-ventilated areas to avoid inhalation and skin contact.

5.2 Disposal and Environmental Considerations

Dispose of unused material and waste as per hazardous chemical regulations.

5.3 Regulatory Status

Flubrotizolam is a controlled research chemical regulated by local laws. It is strictly for research purposes, not for human consumption.

Frequently Asked Questions (FAQs)

1. What is the dosage per Fanax bar?
   0.5 mg of Flubrotizolam.

2. What is the chemical formula?
   C17H12BrFN4S.

3. What effects does Flubrotizolam have?
   Sedation, anxiolysis, muscle relaxation.

4. How is Flubrotizolam used in research?
   CNS pharmacology and benzodiazepine receptor studies.

5. How should Fanax bars be stored?
   Airtight, cool, dry, and dark conditions.

Conclusion

Flubrotizolam 0.5 MG Fanax Bars provide a potent, accurately dosed benzodiazepine research tool ideal for exploring GABAergic CNS mechanisms. Their stable, solid form and precise dosage support rigorous neuropharmacological and behavioral studies.